ABCG2 | ATP-binding cassette sub-family G member 2
 
image/svg+xmlExtracellular space Cytosol Plasma membrane Cytoskeleton Lysosome Endosome Peroxisome ER Golgi Apparatus Nucleus Mitochondrion None Substrate Localization legend

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Sequence Viewer
Gene
Synonyms
ABCP BCRP BCRP1 MXR
Protein Name
ATP-binding cassette sub-family G member 2
UniProt ID
Q9UNQ0 [go to UniProt ] [go to PDBe-KB ]
Ensembl Gene ID
NCBI Gene ID
Molecular Weight
72314
Protein Length
655
Protein Domain
3D Structure
(PDB ID : 5nj3)
Target by Small Molecules
Protein-protein Interaction Database
Gene Expression
Drugs and Diseases
Enzyme Class
-
Catalytic Site
Catalytic Activity
-
Localization
Cell membrane,Mitochondrion membrane;
Function
High-capacity urate exporter functioning in both renal and extrarenal urate excretion. Plays a role in porphyrin homeostasis as it is able to mediates the export of protoporhyrin IX (PPIX) both from mitochondria to cytosol and from cytosol to extracellular space, and cellular export of hemin, and heme. Xenobiotic transporter that may play an important role in the exclusion of xenobiotics from the brain. Appears to play a major role in the multidrug resistance phenotype of several cancer cell lines. Implicated in the efflux of numerous drugs and xenobiotics: mitoxantrone, the photosensitizer pheophorbide, camptothecin, methotrexate, azidothymidine (AZT), and the anthracyclines daunorubicin and doxorubicin.
Gene Ontology
GO:0016021; GO:0031966; GO:0005634; GO:0005886; GO:0005524; GO:0042626; GO:0015232; GO:0042802; GO:0042803; GO:0005215; GO:0008559; GO:0006879; GO:0042493; GO:0055085; GO:0046415
 
Gene Ontology